8-CPT-2Me-cAMP, sodium salt

Mfr.No.	T22014
Description	8-CPT-2Me-cAMP sodium is a sodium salt compound that selectively activates exchange proteins activated by cAMP (Epac). These Epac proteins are cAMP-sensitive guanine nucleotide exchange factors (GEFs) responsible for activating small GTPases Rap1 and Rap2. 8-CPT-2Me-cAMP sodium specifically activates Epac1 with an EC50 value of 2.2 uM, while showing no activation of PKA with an EC50 value greater than 10 uM (1). Additionally, 8-CPT-2Me-cAMP sodium stimulates the Epac-mediated release of calcium ions (Ca2+) in vitro in pancreatic beta-cells (2).
Molecular Formula	C17H16ClN5NaO6PS
Signaling Pathways	Others
Smiles	(Na+).CO(CH)1(CH)2OP((O-))(=O)OC(CH)2O(CH)1n1c(Sc2ccc(Cl)cc2)nc2c(N)ncnc12
Cas Number	634207-53-7
Molecular Weight	507.82
Target	Others

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SKU	Supplier No.	Size	Your price
BHB20411996	T22014	1 mg	$535	Add to Cart
BHB20411996	T22014	5 mg	$2240	Add to Cart
BHB20411996	T22014	500 ?g	$283	Add to Cart